DE69811117T2 - Tetrahydrothiopyran-phenyloxazolidinon-s-oxide - Google Patents
Tetrahydrothiopyran-phenyloxazolidinon-s-oxideInfo
- Publication number
- DE69811117T2 DE69811117T2 DE69811117T DE69811117T DE69811117T2 DE 69811117 T2 DE69811117 T2 DE 69811117T2 DE 69811117 T DE69811117 T DE 69811117T DE 69811117 T DE69811117 T DE 69811117T DE 69811117 T2 DE69811117 T2 DE 69811117T2
- Authority
- DE
- Germany
- Prior art keywords
- phenyloxazolidinone
- tetrahydrothiopyran
- oxide
- dichloromethyl
- fluoro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US6783097P | 1997-12-05 | 1997-12-05 | |
US8949898P | 1998-06-16 | 1998-06-16 | |
US10018598P | 1998-09-14 | 1998-09-14 | |
PCT/US1998/024526 WO1999029688A1 (en) | 1997-12-05 | 1998-11-23 | S-oxide and s,s-dioxide tetrahydrothiopyran phenyloxazolidinones |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69811117D1 DE69811117D1 (de) | 2003-03-06 |
DE69811117T2 true DE69811117T2 (de) | 2003-07-17 |
Family
ID=27371238
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69811117T Expired - Fee Related DE69811117T2 (de) | 1997-12-05 | 1998-11-23 | Tetrahydrothiopyran-phenyloxazolidinon-s-oxide |
Country Status (22)
Country | Link |
---|---|
US (2) | US6083967A (de) |
EP (2) | EP1254906A1 (de) |
JP (1) | JP2001525408A (de) |
KR (1) | KR20010032782A (de) |
CN (2) | CN1532535A (de) |
AT (1) | ATE231859T1 (de) |
AU (2) | AU752454B2 (de) |
BR (1) | BR9814897A (de) |
CA (1) | CA2309026A1 (de) |
DE (1) | DE69811117T2 (de) |
DK (1) | DK1036074T3 (de) |
ES (1) | ES2191985T3 (de) |
HK (1) | HK1032970A1 (de) |
HU (1) | HUP0100558A3 (de) |
ID (1) | ID21450A (de) |
NO (1) | NO316447B1 (de) |
NZ (1) | NZ504930A (de) |
PL (1) | PL340835A1 (de) |
SI (1) | SI1036074T1 (de) |
SK (1) | SK7692000A3 (de) |
TW (2) | TWI239331B (de) |
WO (1) | WO1999029688A1 (de) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6511468B1 (en) | 1997-10-17 | 2003-01-28 | Micro Therapeutics, Inc. | Device and method for controlling injection of liquid embolic composition |
HUP0103082A3 (en) | 1998-06-05 | 2002-12-28 | Astrazeneca Ab | Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them |
MY120189A (en) | 1999-11-04 | 2005-09-30 | Upjohn Co | Sultam and sultone derived oxazolidinones |
DE19962924A1 (de) | 1999-12-24 | 2001-07-05 | Bayer Ag | Substituierte Oxazolidinone und ihre Verwendung |
DE10129725A1 (de) | 2001-06-20 | 2003-01-02 | Bayer Ag | Kombinationstherapie substituierter Oxazolidinone |
AR038536A1 (es) | 2002-02-25 | 2005-01-19 | Upjohn Co | N-aril-2-oxazolidinona-5- carboxamidas y sus derivados |
US7141588B2 (en) | 2002-02-25 | 2006-11-28 | Pfizer, Inc. | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
WO2004014897A1 (en) | 2002-08-12 | 2004-02-19 | Pharmacia & Upjohn Company Llc | N-aryl-2-oxazolidinones and their derivatives |
JP2006509035A (ja) | 2002-11-21 | 2006-03-16 | ファルマシア・アンド・アップジョン・カンパニー・エルエルシー | 抗菌剤としてのn−(4−(ピペラジン−1−イル)−フェニル−2−オキサゾリジノン−5−カルボキサミド誘導体および関連化合物 |
DE10300111A1 (de) | 2003-01-07 | 2004-07-15 | Bayer Healthcare Ag | Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid |
US7304050B2 (en) | 2003-09-16 | 2007-12-04 | Pfizer Inc. | Antibacterial agents |
DE10355461A1 (de) | 2003-11-27 | 2005-06-23 | Bayer Healthcare Ag | Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung |
DE102004062475A1 (de) * | 2004-12-24 | 2006-07-06 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung |
EP1685841A1 (de) | 2005-01-31 | 2006-08-02 | Bayer Health Care Aktiengesellschaft | Prophylaxe und Behandlung von thrombolischen Erkrankungen |
DE102005045518A1 (de) | 2005-09-23 | 2007-03-29 | Bayer Healthcare Ag | 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung |
DE102005047561A1 (de) | 2005-10-04 | 2007-04-05 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung |
DE102005047558A1 (de) * | 2005-10-04 | 2008-02-07 | Bayer Healthcare Ag | Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen |
KR101364400B1 (ko) | 2005-10-04 | 2014-02-17 | 바이엘 인텔렉쳐 프로퍼티 게엠베하 | 5-클로로-n-({(5s)-2-옥소-3-[4-(3-옥소-4-모르폴리닐)-페닐]-1,3-옥사졸리딘-5-일}-메틸)-2-티오펜 카르복사미드의 신규 다형체 및 무정형 형태 |
CN102262066A (zh) * | 2011-06-16 | 2011-11-30 | 董理 | 一种检测单胺氧化酶含量的方法和试剂盒 |
CN104610479B (zh) * | 2013-11-05 | 2017-03-29 | 中国石油化工股份有限公司 | 用于乙烯聚合的负载化茂金属催化剂及其制备方法和应用 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2031921T3 (es) * | 1986-09-03 | 1993-01-01 | Delalande S.A. | Derivados 5-aminoetilados de la oxazolidinona-2, su procedimiento de fabricacion y su aplicacion terapeutica. |
US4885154A (en) * | 1988-03-01 | 1989-12-05 | Alza Corporation | Method for reducing sensitization or irritation in transdermal drug delivery and means therefor |
US5254577A (en) * | 1988-07-29 | 1993-10-19 | The Du Pont Merck Pharmaceutical Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
US5130316A (en) * | 1988-07-29 | 1992-07-14 | Du Pont Merck Pharmaceutical Company | Aminomethyloxooxazlidinyl arylbenzene derivatives useful as antibacterial agents |
US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
JP2669579B2 (ja) * | 1991-10-23 | 1997-10-29 | エーザイ株式会社 | オキサゾリドン誘導体 |
AU667198B2 (en) * | 1991-11-01 | 1996-03-14 | Pharmacia & Upjohn Company | Substituted aryl- and heteroarylphenyloxazolidinones useful as antibacterial agents |
AU670842B2 (en) * | 1992-12-08 | 1996-08-01 | Pharmacia & Upjohn Company | Tropone-substituted phenyloxazolidinone antibacterial agents |
KR100463772B1 (ko) * | 1995-09-01 | 2005-11-09 | 파마시아 앤드 업존 캄파니 엘엘씨 | 4내지8원헤테로사이클릭환에탄소-탄소결합을갖는페닐옥사졸리디논 |
GB9702213D0 (en) * | 1996-02-24 | 1997-03-26 | Zeneca Ltd | Chemical compounds |
-
1998
- 1998-11-20 US US09/196,890 patent/US6083967A/en not_active Expired - Fee Related
- 1998-11-23 AT AT98962811T patent/ATE231859T1/de not_active IP Right Cessation
- 1998-11-23 SI SI9830371T patent/SI1036074T1/xx unknown
- 1998-11-23 HU HU0100558A patent/HUP0100558A3/hu unknown
- 1998-11-23 BR BR9814897-4A patent/BR9814897A/pt not_active Application Discontinuation
- 1998-11-23 CN CNA2004100328277A patent/CN1532535A/zh active Pending
- 1998-11-23 CA CA002309026A patent/CA2309026A1/en not_active Abandoned
- 1998-11-23 AU AU17968/99A patent/AU752454B2/en not_active Ceased
- 1998-11-23 CN CNB988110695A patent/CN1154645C/zh not_active Expired - Fee Related
- 1998-11-23 DE DE69811117T patent/DE69811117T2/de not_active Expired - Fee Related
- 1998-11-23 DK DK98962811T patent/DK1036074T3/da active
- 1998-11-23 EP EP02015566A patent/EP1254906A1/de not_active Withdrawn
- 1998-11-23 KR KR1020007006081A patent/KR20010032782A/ko not_active Application Discontinuation
- 1998-11-23 WO PCT/US1998/024526 patent/WO1999029688A1/en active Search and Examination
- 1998-11-23 PL PL98340835A patent/PL340835A1/xx unknown
- 1998-11-23 ES ES98962811T patent/ES2191985T3/es not_active Expired - Lifetime
- 1998-11-23 EP EP98962811A patent/EP1036074B1/de not_active Expired - Lifetime
- 1998-11-23 JP JP2000524282A patent/JP2001525408A/ja active Pending
- 1998-11-23 SK SK769-2000A patent/SK7692000A3/sk unknown
- 1998-11-23 NZ NZ504930A patent/NZ504930A/en unknown
- 1998-11-26 ID IDP981545A patent/ID21450A/id unknown
- 1998-12-04 TW TW092121194A patent/TWI239331B/zh not_active IP Right Cessation
- 1998-12-04 TW TW087120185A patent/TW553942B/zh not_active IP Right Cessation
-
1999
- 1999-11-05 US US09/434,911 patent/US6265178B1/en not_active Expired - Fee Related
-
2000
- 2000-06-02 NO NO20002834A patent/NO316447B1/no unknown
-
2001
- 2001-05-24 HK HK01103598A patent/HK1032970A1/xx not_active IP Right Cessation
-
2002
- 2002-09-16 AU AU2002301031A patent/AU2002301031B2/en not_active Ceased
Also Published As
Publication number | Publication date |
---|---|
ID21450A (id) | 1999-06-10 |
EP1036074A1 (de) | 2000-09-20 |
PL340835A1 (en) | 2001-02-26 |
TWI239331B (en) | 2005-09-11 |
DK1036074T3 (da) | 2003-06-23 |
HUP0100558A3 (en) | 2002-08-28 |
JP2001525408A (ja) | 2001-12-11 |
CN1154645C (zh) | 2004-06-23 |
ATE231859T1 (de) | 2003-02-15 |
US6265178B1 (en) | 2001-07-24 |
NZ504930A (en) | 2002-05-31 |
CN1532535A (zh) | 2004-09-29 |
CN1278817A (zh) | 2001-01-03 |
AU1796899A (en) | 1999-06-28 |
CA2309026A1 (en) | 1999-06-17 |
NO316447B1 (no) | 2004-01-26 |
AU2002301031B2 (en) | 2005-08-25 |
SI1036074T1 (en) | 2003-08-31 |
EP1036074B1 (de) | 2003-01-29 |
HK1032970A1 (en) | 2001-08-10 |
NO20002834L (no) | 2000-07-21 |
TW200307673A (en) | 2003-12-16 |
SK7692000A3 (en) | 2001-03-12 |
NO20002834D0 (no) | 2000-06-02 |
KR20010032782A (ko) | 2001-04-25 |
DE69811117D1 (de) | 2003-03-06 |
ES2191985T3 (es) | 2003-09-16 |
AU752454B2 (en) | 2002-09-19 |
HUP0100558A2 (hu) | 2002-05-29 |
EP1254906A1 (de) | 2002-11-06 |
WO1999029688A1 (en) | 1999-06-17 |
BR9814897A (pt) | 2000-10-03 |
TW553942B (en) | 2003-09-21 |
US6083967A (en) | 2000-07-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |