DE69811117D1 - Tetrahydrothiopyran-phenyloxazolidinon-s-oxide - Google Patents
Tetrahydrothiopyran-phenyloxazolidinon-s-oxideInfo
- Publication number
- DE69811117D1 DE69811117D1 DE69811117T DE69811117T DE69811117D1 DE 69811117 D1 DE69811117 D1 DE 69811117D1 DE 69811117 T DE69811117 T DE 69811117T DE 69811117 T DE69811117 T DE 69811117T DE 69811117 D1 DE69811117 D1 DE 69811117D1
- Authority
- DE
- Germany
- Prior art keywords
- phenyloxazolidinone
- tetrahydrothiopyran
- oxide
- dichloromethyl
- fluoro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US6783097P | 1997-12-05 | 1997-12-05 | |
US8949898P | 1998-06-16 | 1998-06-16 | |
US10018598P | 1998-09-14 | 1998-09-14 | |
PCT/US1998/024526 WO1999029688A1 (en) | 1997-12-05 | 1998-11-23 | S-oxide and s,s-dioxide tetrahydrothiopyran phenyloxazolidinones |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69811117D1 true DE69811117D1 (de) | 2003-03-06 |
DE69811117T2 DE69811117T2 (de) | 2003-07-17 |
Family
ID=27371238
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69811117T Expired - Fee Related DE69811117T2 (de) | 1997-12-05 | 1998-11-23 | Tetrahydrothiopyran-phenyloxazolidinon-s-oxide |
Country Status (22)
Country | Link |
---|---|
US (2) | US6083967A (de) |
EP (2) | EP1254906A1 (de) |
JP (1) | JP2001525408A (de) |
KR (1) | KR20010032782A (de) |
CN (2) | CN1154645C (de) |
AT (1) | ATE231859T1 (de) |
AU (2) | AU752454B2 (de) |
BR (1) | BR9814897A (de) |
CA (1) | CA2309026A1 (de) |
DE (1) | DE69811117T2 (de) |
DK (1) | DK1036074T3 (de) |
ES (1) | ES2191985T3 (de) |
HK (1) | HK1032970A1 (de) |
HU (1) | HUP0100558A3 (de) |
ID (1) | ID21450A (de) |
NO (1) | NO316447B1 (de) |
NZ (1) | NZ504930A (de) |
PL (1) | PL340835A1 (de) |
SI (1) | SI1036074T1 (de) |
SK (1) | SK7692000A3 (de) |
TW (2) | TWI239331B (de) |
WO (1) | WO1999029688A1 (de) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6511468B1 (en) * | 1997-10-17 | 2003-01-28 | Micro Therapeutics, Inc. | Device and method for controlling injection of liquid embolic composition |
MXPA00011536A (es) | 1998-06-05 | 2002-10-17 | Astrazeneca Ab | Derivados de oxazolidinona, proceso para su preparacion y composiciones farmaceuticas que las contienen. |
MY120189A (en) * | 1999-11-04 | 2005-09-30 | Upjohn Co | Sultam and sultone derived oxazolidinones |
DE19962924A1 (de) | 1999-12-24 | 2001-07-05 | Bayer Ag | Substituierte Oxazolidinone und ihre Verwendung |
DE10129725A1 (de) | 2001-06-20 | 2003-01-02 | Bayer Ag | Kombinationstherapie substituierter Oxazolidinone |
US7141588B2 (en) | 2002-02-25 | 2006-11-28 | Pfizer, Inc. | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
AR038536A1 (es) | 2002-02-25 | 2005-01-19 | Upjohn Co | N-aril-2-oxazolidinona-5- carboxamidas y sus derivados |
AU2003259159A1 (en) | 2002-08-12 | 2004-02-25 | Pharmacia & Upjohn Company Llc | N-aryl-2-oxazolidinones and their derivatives |
US7141570B2 (en) | 2002-11-21 | 2006-11-28 | Pharmacia & Upjohn Company | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
DE10300111A1 (de) | 2003-01-07 | 2004-07-15 | Bayer Healthcare Ag | Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid |
US7304050B2 (en) | 2003-09-16 | 2007-12-04 | Pfizer Inc. | Antibacterial agents |
DE10355461A1 (de) | 2003-11-27 | 2005-06-23 | Bayer Healthcare Ag | Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung |
DE102004062475A1 (de) * | 2004-12-24 | 2006-07-06 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung |
EP1685841A1 (de) | 2005-01-31 | 2006-08-02 | Bayer Health Care Aktiengesellschaft | Prophylaxe und Behandlung von thrombolischen Erkrankungen |
DE102005045518A1 (de) | 2005-09-23 | 2007-03-29 | Bayer Healthcare Ag | 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung |
DE102005047561A1 (de) | 2005-10-04 | 2007-04-05 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung |
AU2006299126B2 (en) | 2005-10-04 | 2012-06-28 | Bayer Intellectual Property Gmbh | Novel polymorphous form and the amorphous form of 5-chloro-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidine-5-yl}-methyl)-2-thiophene carboxamide |
DE102005047558A1 (de) * | 2005-10-04 | 2008-02-07 | Bayer Healthcare Ag | Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen |
CN102262066A (zh) * | 2011-06-16 | 2011-11-30 | 董理 | 一种检测单胺氧化酶含量的方法和试剂盒 |
CN104610479B (zh) * | 2013-11-05 | 2017-03-29 | 中国石油化工股份有限公司 | 用于乙烯聚合的负载化茂金属催化剂及其制备方法和应用 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4897409A (en) * | 1986-09-03 | 1990-01-30 | Delalande S.A. | 5-aminoethyloxazolidin-2-one derivatives |
US4885154A (en) * | 1988-03-01 | 1989-12-05 | Alza Corporation | Method for reducing sensitization or irritation in transdermal drug delivery and means therefor |
US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
US5254577A (en) * | 1988-07-29 | 1993-10-19 | The Du Pont Merck Pharmaceutical Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
US5130316A (en) * | 1988-07-29 | 1992-07-14 | Du Pont Merck Pharmaceutical Company | Aminomethyloxooxazlidinyl arylbenzene derivatives useful as antibacterial agents |
JP2669579B2 (ja) * | 1991-10-23 | 1997-10-29 | エーザイ株式会社 | オキサゾリドン誘導体 |
KR100257418B1 (ko) * | 1991-11-01 | 2000-05-15 | 로렌스 티. 마이젠헬더 | 치환된 아릴-및 헤테로아릴-페닐옥사졸리디논 |
CA2147753C (en) * | 1992-12-08 | 2004-08-03 | Michael Robert Barbachyn | Tropone-substituted phenyloxazolidinone antibacterial agents |
BR9610474A (pt) * | 1995-09-01 | 1999-03-02 | Upjohn Co | Feniloxazolidinonas tendo uma ligação c-c a anéis heterocíclicos com 4-8 membros |
GB9702213D0 (en) * | 1996-02-24 | 1997-03-26 | Zeneca Ltd | Chemical compounds |
-
1998
- 1998-11-20 US US09/196,890 patent/US6083967A/en not_active Expired - Fee Related
- 1998-11-23 ES ES98962811T patent/ES2191985T3/es not_active Expired - Lifetime
- 1998-11-23 EP EP02015566A patent/EP1254906A1/de not_active Withdrawn
- 1998-11-23 WO PCT/US1998/024526 patent/WO1999029688A1/en active Search and Examination
- 1998-11-23 SI SI9830371T patent/SI1036074T1/xx unknown
- 1998-11-23 NZ NZ504930A patent/NZ504930A/en unknown
- 1998-11-23 SK SK769-2000A patent/SK7692000A3/sk unknown
- 1998-11-23 BR BR9814897-4A patent/BR9814897A/pt not_active Application Discontinuation
- 1998-11-23 EP EP98962811A patent/EP1036074B1/de not_active Expired - Lifetime
- 1998-11-23 CA CA002309026A patent/CA2309026A1/en not_active Abandoned
- 1998-11-23 KR KR1020007006081A patent/KR20010032782A/ko not_active Application Discontinuation
- 1998-11-23 AU AU17968/99A patent/AU752454B2/en not_active Ceased
- 1998-11-23 CN CNB988110695A patent/CN1154645C/zh not_active Expired - Fee Related
- 1998-11-23 AT AT98962811T patent/ATE231859T1/de not_active IP Right Cessation
- 1998-11-23 HU HU0100558A patent/HUP0100558A3/hu unknown
- 1998-11-23 CN CNA2004100328277A patent/CN1532535A/zh active Pending
- 1998-11-23 DE DE69811117T patent/DE69811117T2/de not_active Expired - Fee Related
- 1998-11-23 PL PL98340835A patent/PL340835A1/xx unknown
- 1998-11-23 DK DK98962811T patent/DK1036074T3/da active
- 1998-11-23 JP JP2000524282A patent/JP2001525408A/ja active Pending
- 1998-11-26 ID IDP981545A patent/ID21450A/id unknown
- 1998-12-04 TW TW092121194A patent/TWI239331B/zh not_active IP Right Cessation
- 1998-12-04 TW TW087120185A patent/TW553942B/zh not_active IP Right Cessation
-
1999
- 1999-11-05 US US09/434,911 patent/US6265178B1/en not_active Expired - Fee Related
-
2000
- 2000-06-02 NO NO20002834A patent/NO316447B1/no unknown
-
2001
- 2001-05-24 HK HK01103598A patent/HK1032970A1/xx not_active IP Right Cessation
-
2002
- 2002-09-16 AU AU2002301031A patent/AU2002301031B2/en not_active Ceased
Also Published As
Publication number | Publication date |
---|---|
SI1036074T1 (en) | 2003-08-31 |
DE69811117T2 (de) | 2003-07-17 |
ATE231859T1 (de) | 2003-02-15 |
NO316447B1 (no) | 2004-01-26 |
CN1278817A (zh) | 2001-01-03 |
AU1796899A (en) | 1999-06-28 |
US6083967A (en) | 2000-07-04 |
HK1032970A1 (en) | 2001-08-10 |
HUP0100558A3 (en) | 2002-08-28 |
EP1254906A1 (de) | 2002-11-06 |
BR9814897A (pt) | 2000-10-03 |
WO1999029688A1 (en) | 1999-06-17 |
NO20002834L (no) | 2000-07-21 |
CN1154645C (zh) | 2004-06-23 |
EP1036074B1 (de) | 2003-01-29 |
HUP0100558A2 (hu) | 2002-05-29 |
PL340835A1 (en) | 2001-02-26 |
TW553942B (en) | 2003-09-21 |
ES2191985T3 (es) | 2003-09-16 |
CA2309026A1 (en) | 1999-06-17 |
NZ504930A (en) | 2002-05-31 |
US6265178B1 (en) | 2001-07-24 |
TWI239331B (en) | 2005-09-11 |
CN1532535A (zh) | 2004-09-29 |
AU2002301031B2 (en) | 2005-08-25 |
KR20010032782A (ko) | 2001-04-25 |
NO20002834D0 (no) | 2000-06-02 |
JP2001525408A (ja) | 2001-12-11 |
DK1036074T3 (da) | 2003-06-23 |
TW200307673A (en) | 2003-12-16 |
ID21450A (id) | 1999-06-10 |
AU752454B2 (en) | 2002-09-19 |
EP1036074A1 (de) | 2000-09-20 |
SK7692000A3 (en) | 2001-03-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |