DE69616366T2 - Phenyloxazolidinone mit einer c-c-bindung zu 4-8 gliedrigen heterocyclen - Google Patents

Phenyloxazolidinone mit einer c-c-bindung zu 4-8 gliedrigen heterocyclen

Info

Publication number
DE69616366T2
DE69616366T2 DE69616366T DE69616366T DE69616366T2 DE 69616366 T2 DE69616366 T2 DE 69616366T2 DE 69616366 T DE69616366 T DE 69616366T DE 69616366 T DE69616366 T DE 69616366T DE 69616366 T2 DE69616366 T2 DE 69616366T2
Authority
DE
Germany
Prior art keywords
alkyl
halo
aryl
methyl
substd
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69616366T
Other languages
English (en)
Other versions
DE69616366D1 (de
Inventor
K Hutchinson
D Ennis
L Hoffman
C Thomas
Toni-Jo Poel
Robert Barbachyn
J Brickner
J Anderson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co
Original Assignee
Pharmacia and Upjohn Co
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia and Upjohn Co, Upjohn Co filed Critical Pharmacia and Upjohn Co
Application granted granted Critical
Publication of DE69616366D1 publication Critical patent/DE69616366D1/de
Publication of DE69616366T2 publication Critical patent/DE69616366T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
DE69616366T 1995-09-01 1996-08-13 Phenyloxazolidinone mit einer c-c-bindung zu 4-8 gliedrigen heterocyclen Expired - Fee Related DE69616366T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US314995P 1995-09-01 1995-09-01
PCT/US1996/012766 WO1997009328A1 (en) 1995-09-01 1996-08-13 Phenyloxazolidinones having a c-c bond to 4-8 membered heterocyclic rings

Publications (2)

Publication Number Publication Date
DE69616366D1 DE69616366D1 (de) 2001-11-29
DE69616366T2 true DE69616366T2 (de) 2002-07-04

Family

ID=21704418

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69616366T Expired - Fee Related DE69616366T2 (de) 1995-09-01 1996-08-13 Phenyloxazolidinone mit einer c-c-bindung zu 4-8 gliedrigen heterocyclen

Country Status (27)

Country Link
US (7) US5968962A (de)
EP (1) EP0856002B1 (de)
JP (1) JPH11512386A (de)
KR (1) KR100463772B1 (de)
CN (1) CN1072222C (de)
AT (1) ATE207487T1 (de)
AU (1) AU716493B2 (de)
BR (1) BR9610474A (de)
CA (1) CA2228647A1 (de)
CZ (1) CZ49398A3 (de)
DE (1) DE69616366T2 (de)
DK (1) DK0856002T3 (de)
ES (1) ES2165516T3 (de)
FI (1) FI980452A0 (de)
HK (1) HK1014946A1 (de)
HU (1) HUP9901979A3 (de)
MX (1) MX9801578A (de)
NO (1) NO311520B1 (de)
NZ (1) NZ315469A (de)
PL (1) PL186524B1 (de)
PT (1) PT856002E (de)
RU (1) RU2175324C2 (de)
SK (1) SK283487B6 (de)
TW (1) TW419468B (de)
UA (1) UA52620C2 (de)
WO (1) WO1997009328A1 (de)
ZA (1) ZA966935B (de)

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AU2003259159A1 (en) * 2002-08-12 2004-02-25 Pharmacia & Upjohn Company Llc N-aryl-2-oxazolidinones and their derivatives
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JP5161070B2 (ja) 2006-03-31 2013-03-13 財団法人乙卯研究所 ヘテロ環を有する新規化合物
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TW202317534A (zh) 2021-06-16 2023-05-01 美商西建公司 用於治療神經退化性疾病之含羧酸吖丁啶基化合物
CN115724823B (zh) * 2021-08-27 2023-11-24 中国科学院大连化学物理研究所 一种制备二氢噻吩衍生物的方法

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Also Published As

Publication number Publication date
AU716493B2 (en) 2000-02-24
CA2228647A1 (en) 1997-03-13
KR100463772B1 (ko) 2005-11-09
BR9610474A (pt) 1999-03-02
FI980452A (fi) 1998-02-27
DK0856002T3 (da) 2002-02-11
JPH11512386A (ja) 1999-10-26
NO980855D0 (no) 1998-02-27
RU2175324C2 (ru) 2001-10-27
NO980855L (no) 1998-04-30
EP0856002B1 (de) 2001-10-24
KR19990044238A (ko) 1999-06-25
UA52620C2 (uk) 2003-01-15
US6051716A (en) 2000-04-18
DE69616366D1 (de) 2001-11-29
FI980452A0 (fi) 1998-02-27
ES2165516T3 (es) 2002-03-16
AU6718196A (en) 1997-03-27
HUP9901979A3 (en) 2000-03-28
PL186524B1 (pl) 2004-01-30
TW419468B (en) 2001-01-21
CZ49398A3 (cs) 1998-08-12
US6358942B1 (en) 2002-03-19
US6043266A (en) 2000-03-28
US20050054683A1 (en) 2005-03-10
CN1197457A (zh) 1998-10-28
US6313307B1 (en) 2001-11-06
ATE207487T1 (de) 2001-11-15
MX9801578A (es) 1998-08-30
EP0856002A1 (de) 1998-08-05
NO311520B1 (no) 2001-12-03
US6166056A (en) 2000-12-26
ZA966935B (en) 1998-02-16
PL325152A1 (en) 1998-07-06
SK283487B6 (sk) 2003-08-05
NZ315469A (en) 2000-01-28
CN1072222C (zh) 2001-10-03
HUP9901979A2 (hu) 2000-02-28
SK19598A3 (en) 1998-11-04
WO1997009328A1 (en) 1997-03-13
PT856002E (pt) 2002-04-29
HK1014946A1 (en) 1999-10-08
US5968962A (en) 1999-10-19

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