DE69216251T2 - Substituierte aryl- und heteroaryl-phenyloxazolidinone - Google Patents

Substituierte aryl- und heteroaryl-phenyloxazolidinone

Info

Publication number
DE69216251T2
DE69216251T2 DE69216251T DE69216251T DE69216251T2 DE 69216251 T2 DE69216251 T2 DE 69216251T2 DE 69216251 T DE69216251 T DE 69216251T DE 69216251 T DE69216251 T DE 69216251T DE 69216251 T2 DE69216251 T2 DE 69216251T2
Authority
DE
Germany
Prior art keywords
substituted aryl
heteroaryl
phenyloxazolidinone
heteroarylphenyloxazolidinones
oxazolidinones
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69216251T
Other languages
English (en)
Other versions
DE69216251D1 (en
Inventor
Michael Barbachyn
Steven Brickner
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co
Original Assignee
Pharmacia and Upjohn Co
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia and Upjohn Co, Upjohn Co filed Critical Pharmacia and Upjohn Co
Application granted granted Critical
Publication of DE69216251D1 publication Critical patent/DE69216251D1/de
Publication of DE69216251T2 publication Critical patent/DE69216251T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
DE69216251T 1991-11-01 1992-10-05 Substituierte aryl- und heteroaryl-phenyloxazolidinone Expired - Fee Related DE69216251T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US78610791A 1991-11-01 1991-11-01
US83121392A 1992-02-07 1992-02-07
PCT/US1992/008267 WO1993009103A1 (en) 1991-11-01 1992-10-05 Substituted aryl- and heteroarylphenyloxazolidinones useful as antibacterial agents

Publications (2)

Publication Number Publication Date
DE69216251D1 DE69216251D1 (en) 1997-02-06
DE69216251T2 true DE69216251T2 (de) 1997-05-15

Family

ID=27120493

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69216251T Expired - Fee Related DE69216251T2 (de) 1991-11-01 1992-10-05 Substituierte aryl- und heteroaryl-phenyloxazolidinone

Country Status (11)

Country Link
US (6) US5565571A (de)
EP (1) EP0610265B1 (de)
JP (1) JP3176626B2 (de)
KR (1) KR100257418B1 (de)
AT (1) ATE146783T1 (de)
AU (1) AU667198B2 (de)
CA (1) CA2119556C (de)
DE (1) DE69216251T2 (de)
DK (1) DK0610265T3 (de)
GR (1) GR3022340T3 (de)
WO (1) WO1993009103A1 (de)

Families Citing this family (143)

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AU2689892A (en) 1993-06-07
WO1993009103A1 (en) 1993-05-13
CA2119556A1 (en) 1993-05-13
CA2119556C (en) 2004-07-06
US5565571A (en) 1996-10-15
US5654435A (en) 1997-08-05
JPH07500603A (ja) 1995-01-19
US5929248A (en) 1999-07-27
AU667198B2 (en) 1996-03-14
KR100257418B1 (ko) 2000-05-15
DK0610265T3 (da) 1997-06-09
EP0610265B1 (de) 1996-12-27
JP3176626B2 (ja) 2001-06-18
US5756732A (en) 1998-05-26
ATE146783T1 (de) 1997-01-15
DE69216251D1 (en) 1997-02-06
US5801246A (en) 1998-09-01
US5654428A (en) 1997-08-05
EP0610265A1 (de) 1994-08-17

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